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Re: Receptor Infinities » Brainbeard

Posted by Conundrum on May 24, 2010, at 20:54:09

In reply to Receptor Infinities, posted by Brainbeard on May 24, 2010, at 13:28:27

Nice topic title. Here is the search results for Nortriptyline for some reason there are two entries:

http://pdsp.med.unc.edu/pdsp.php?knowID=&kiKey=&receptorDD=&receptor=&speciesDD=&species=&sourcesDD=&source=&hotLigandDD=&hotLigand=&testDDRadio=testDDRadio&testLigandDD=2060&testLigand=&referenceDD=&reference=&KiGreater=&KiLess=&kiAllRadio=all&doQuery=Submit+Query

and

http://pdsp.med.unc.edu/pdsp.php?knowID=&kiKey=&receptorDD=&receptor=&speciesDD=&species=&sourcesDD=&source=&hotLigandDD=&hotLigand=&testDDRadio=testDDRadio&testLigandDD=7404&testLigand=&referenceDD=&reference=&KiGreater=&KiLess=&kiAllRadio=all&doQuery=Submit+Query

Amitriptyline:
http://pdsp.med.unc.edu/pdsp.php?knowID=&kiKey=&recDDRadio=recDDRadio&receptorDD=&receptor=&speciesDD=&species=&sourcesDD=&source=&hotLigandDD=&hotLigand=&testDDRadio=testDDRadio&testLigandDD=788&testLigand=&referenceDD=&reference=&KiGreater=&KiLess=&kiAllRadio=all&doQuery=Submit+Query

Desipramine:
http://pdsp.med.unc.edu/pdsp.php?knowID=&kiKey=&receptorDD=&receptor=&speciesDD=&species=&sourcesDD=&source=&hotLigandDD=&hotLigand=&testDDRadio=testDDRadio&testLigandDD=1197&testLigand=&referenceDD=&reference=&KiGreater=&KiLess=&kiAllRadio=all&doQuery=Submit+Query

Imipramine:
http://pdsp.med.unc.edu/pdsp.php?knowID=&kiKey=&receptorDD=&receptor=&speciesDD=&species=&sourcesDD=&source=&hotLigandDD=&hotLigand=&testDDRadio=testDDRadio&testLigandDD=1622&testLigand=&referenceDD=&reference=&KiGreater=&KiLess=&kiAllRadio=all&doQuery=Submit+Query


It would be nice to know if these drugs were antagonists or inverse agonists at the receptors they block. So it looks like nortriptyline is definitely "dirtier" than desipramine. It has the benefit of more 5HT2A/C antagonism and the boon of anticholinergic and anti-histaminergic actions. Desipramine is almost pure noradrenline. Good if you just need NE, if you need any antagonism probably would have to add Remeron or some antipyschotic at a low dose. Nortriptyline will be more sedating and could cause lethargy and weight gain and desipramine should be activating, and may cause tachyardia. But I guess you all knew that.

Almost forgot Protriptyline not much on that:

http://pdsp.med.unc.edu/pdsp.php?knowID=&kiKey=&receptorDD=&receptor=&speciesDD=&species=&sourcesDD=&source=&hotLigandDD=&hotLigand=&testDDRadio=testDDRadio&testLigandDD=2268&testLigand=&referenceDD=&reference=&KiGreater=&KiLess=&kiAllRadio=all&doQuery=Submit+Query

For a more visual comparison check this out:

http://www.mindandmuscle.net/forum/index.php?showtopic=38276&pid=552949&mode=threaded&show=&st=0


Post-SSRI syndrome: iatrogenic anhedonia, memory and concentration problems, sexual dysfunction. [NOTE no sadness or anxiety]
Location:USA
Currently taking 25mg Lamictal.

 

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poster:Conundrum thread:943541
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